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中间体产品目录Intermediates:

NO.

PRODUCT NAME

CAS RN.

Agomelatine

1

7-methoxy-1-tetralone

6836-19-7

2

7-Methoxy-1-naphthylacetonitrile

138113-08-3

3

2-(7-Methoxy-1-naphthyl)ethylamine hydrochloride

139525-77-2

Amisulpride

1

4-Amino-5-ethylsulfonyl-2-methoxybenzoic acid

71675-87-1

Aprepitant

1

(R)-1-[3,5-Bis(trifluoromethyl)phenyl]ethanol

127852-28-2

Asenapine Maleate

1

2-(5-chloro-2-phenoxyphenyl)acetic acid

70958-20-2

2

5-chloro-2,3,3a,12b-tetrahydro-2-methyl-1H-Dibenz [2,3:6,7]oxepino[4,5-c]pyrrol-1-one (Cis-Trans mixture)

N/A

3

11-Chloro-2,3-dihydro-2-methyl-1H-dibenz[2,3:6,7]oxepino[4,5-c]pyrrol-1-one

1012884-46-6

4

trans-(+/-)-11-Chloro-2,3,3a,12b-tetrahydro-2-methyl-1H-dibenz[2,3:6,7]oxepino[4,5-c]pyrrol-1-one

129385-59-7

Atazanavir Sulfate

1

Moc-L-tert-Leucine

162537-11-3

2

(2R,3S)-3-(tert-Butoxycarbonyl)amino-1,2-epoxy-4-phenylbutane

98760-08-8

3

L-tert-Leucine

20859-02-3

4

2-[(2S,3S)-3-[[(1,1-Dimethylethoxy)carbonyl]amino]-2-hydroxy-4-phenylbutyl]-2-[[4-(2-pyridinyl)phenyl]methyl]hydrazinecarboxylic acid tert-butyl ester

198904-86-8

5

tert-Butyl 2-(4-(pyridin-2-yl)benzyl)hydrazinecarboxylate

198904-85-7

Baricitinib

1

[4-(1H-Pyrazol-4-yl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl]methyl pivalate

1146629-77-7

Bazedoxifene Acetate

1

3-Methyl-5-(phenylmethoxy)-2-[4-(phenylmethoxy)phenyl]-1H-indole

198479-63-9

2

1-(2-(4-(Chloromethyl)phenoxy)ethyl)azepane hydrochloride

223251-25-0

3

1-[4-(2-(Azepan-1-yl)ethoxy)benzyl]-5-(benzyloxy)-2-(4-(benzyloxy)phenyl)-3-methyl-1H-indole

198480-21-6

Brexpiprazole

1

1-benzo[b]thien-4-yl-piperazine hydrochloride 

913614-18-3

2

7-hydroxy-2(1H)-quinolinone 

70500-72-0

3

4-Chlorobenzothiophene

66490-33-3

4

4-Bromobenzo[b]thiophene

5118-13-8

5

1-benzo[b]thien-4-yl-piperazine

846038-18-4

6

7-Hydroxy carbostyril

22246-18-0

7

7-(4-Chlorobutoxy)-1H-quinolin-2-one

913613-82-8

Brivaracetam

1

(R)-4-Propyldihydrofuran-2(3H)-one

63095-51-2

2

L-2-Aminobutanamide hydrochloride

7682-20-4

Cangrelor

1

N-[2-(Methylthio)ethyl]-2-[(3,3,3-trifluoropropyl)thio]adenosine

163706-58-9

Chloropromazine

1

3-Dimethylaminopropylchloride hydrochloride

5407-04-5

2

2-Chlorophenothiazine

92-39-7

3

(+)-2,2'-Isopropylidenebis[(4R)-4-phenyl-2-oxazoline]

150529-93-4

Crizotinib

1

(S)-1-(2,6-Dichloro-3-fluorophenyl)ethanol

877397-65-4

2

tert-Butyl 4-[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazol-1-yl]piperidine-1-carboxylate

877399-74-1

3

[5-Bromo-3-[(1R)-(2,6-dichloro-3-fluorophenyl)ethoxy]pyridin-2-yl]amine

877399-00-3

Dapoxetine Hydrochloride

1

(S)-3-Amino-3-phenyl-1-propanol hydrochloride

936499-93-3

Dolutegravir

1

(R)-3-amino-1-butanol

61477-40-5

D-Cycloserine

1

3-Chloro-D-alanine methyl ester hydrochloride

112346-82-4

Ertugliflozin

1

2,3,4,6-tetra-O-benzyl-D-glucopyranose

4132-28-9

Etizolam

1

2-Amino-3-(2-chlorobenzoyl)-5-ethylthiophene

50508-60-6

2

2-(2-Chloroacetamido)-3-(o-chlorobenzoyl)-5-ethylthiophene

50508-89-9

3

2-(Aminoacetamido)-3-(2-chlorobenzoyl)-5-ethylthiophene

50509-09-6

4

N-[3-(2-Chlorobenzoyl)-5-ethyl-2-thienyl]-1,3-dihydro-1,3-dioxo-2H-isoindole-2-acetamide

42753-80-0

5

5-(2-Chlorophenyl)-7-ethyl-1,3-dihydro-2H-thieno[2,3-e]-1,4-diazepin-2-one

33671-37-3

6

5-(2-Chlorophenyl)-7-ethyl-1,3-dihydro-2H-thieno[2,3-e]-1,4-diazepine-2-thione

40054-40-8

Fluvastatin

1

tert-Butyl (E)-7-[3'-(4''-fluorophenyl)-1'-methylethyl-indol-2'-yl]-3-hydroxy-5-oxo-6-heptenoate

375846-25-6

Gadobutrol

1

Cyclen

294-90-6

Gemcitabine

1

2-deoxy-2,2-difluoro-D-erythro-pentofuranos-1-ulose-3,5-dibenzoate

122111-01-7

2

2-Deoxy-2,2-difluoro-D-erythro-pentofuranose-3,5-dibenzoate-1-methanesulfonate

122111-11-9

Ibrutinib

1

(R)-3-(4-Phenoxyphenyl)-1-(piperidin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine

1022150-12-4

2

3-(4-Phenoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine

330786-24-8

3

(S)-1-Boc-3-hydroxypiperidine

143900-44-1

 

 

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